Now reading Entry 010 / 102 Last revised Jan 22, 2026 28 sources 2 comparisons Methodology →
A specimen of the Metabolic drawer Drawer A · Metabolic

Cagrilintide

Investigational

A long-acting amylin analog developed by Novo Nordisk for weight management. Studied in Phase 3 trials as CagriSema (combination with semaglutide). The Phase 3 REDEFINE 1 trial showed -20.4% weight loss with cagrilintide-semaglutide versus -3.0% with placebo at 68 weeks.

AM833 · NN9838

Research evidence
High

18 human studies

Preclinical
36%
Clinical
64%

Based on 28 cited sources

Evidence Score70/100
Emerging / moderate
Research Depth78/100
Mechanism84/100
Plausibility89/100
Global Coverage57/100
Community Experience26/100
Effectiveness84/100

clinically demonstrated · high confidence

Demonstrated effect magnitude — not a recommendation or safety claim.

Research Depth: multiple large placebo-controlled RCTs incl. Phase 3 REDEFINE 1 (n=3,417) and REDEFINE 2, total human N well over 1,000, no published meta-analysis yet. Mechanism: amylin AMY1/2/3 receptors named with binding + functional confirmation and characterized satiety pathway. Plausibility: full mechanism to weight-loss outcome chain supported, coherent with amylin biology and same-class pramlintide. Global Coverage: international multi-country trials but single sponsor (Novo Nordisk) and FDA review pending, limiting independence. Community Experience: trial-only, near-negligible real-world usage signal. Effectiveness basis clinical: REDEFINE 1 (NCT05567796) showed -20.4% weight loss with cagrilintide-semaglutide versus -3.0% with placebo at 68 weeks. Reconciliation (2026-06-27): citation sweep corrected REDEFINE 1 from "~22.7% with head-to-head superiority over semaglutide" to "-20.4% vs -3.0% placebo" — a placebo-controlled (not head-to-head) result; Effectiveness lowered 93 -> 84 (E4 drops from head-to-head-superiority to placebo-superiority; large magnitude E1/E2 retained). Evidence axis unchanged (trial counts/tiers and mechanism intact).

Scored May 2026 How we rate →
Evidence Level
high
Not approved for human use by any regulatory agency
Limited human clinical trial data
Consult a healthcare provider before use
Not FDA Approved WADA Prohibited
Identity
SCALE · 1:1 N-TERMINUS C-TERMINUS 37 AA · ~4,200 Da
Also Known As
AM833 • NN9838
Class
Acylated amylin analog
Length
37 amino acids
Mol. weight
~4,200 Da
Sequence
Modified human amylin with amino acid substitutions + C18 fatty acid acylation
Molecular Structure
K
C
N
T
A
T
C
A
T
Q
R
L
A
N
F
L
V
H
S
S
N
N
F
G
A
I
L
S
S
T
N
V
G
S
N
T
Y
Hydrophobic
Polar
Positive
Negative

Cagrilintide is a long-acting amylin analog that acts through distinct and complementary pathways to GLP-1 agonists. Human clinical trial data supports its efficacy for weight management.

How It Works (Simplified)

Cagrilintide mimics amylin, a hormone co-secreted with insulin that signals satiety through different brain pathways than GLP-1:

Brainstem Satiety

Activates amylin receptors in the area postrema, sending powerful “full” signals to the brain through a different pathway than GLP-1.

Leptin Sensitization

Restores responsiveness to leptin, the body’s natural “stop eating” hormone that becomes impaired in obesity.

Gastric Slowing

Delays gastric emptying, prolonging feelings of fullness and preventing rapid blood sugar spikes after meals.

Glucagon Suppression

Reduces postprandial glucagon release, helping control blood sugar in diabetes without directly stimulating insulin.

Key Research: Lau DCW et al. (2021) demonstrated -10.8% weight loss with cagrilintide 4.5 mg monotherapy in Phase 2 RCT. PMID:34798060

Important Limitations

  • Cagrilintide is an investigational compound with no regulatory approvals
  • All efficacy data from Phase 1b and Phase 2 trials; Phase 3 results pending
  • No long-term safety data beyond 1 year
  • No cardiovascular outcomes data (REDEFINE CVOT ongoing, results 2029)
  • All clinical trials sponsored by Novo Nordisk (developer)
  • Not available outside of clinical trials as of January 2026

Research Tools

i. Amylin Receptor Signaling · Satiety
CagrilintideAMY1/2/3 receptors (area postrema)cAMP signalingSatiety neuronsReduced food intake
ii. Leptin Sensitization Pathway · Metabolic
CagrilintideAmylin receptor activationHypothalamic circuitsRestored leptin responsiveness
Mechanism Amylin receptor (AMY1/2/3) agonism in area postrema triggering satiety signaling
Established 8 direct studies
Benefit shown to reduce appetite and food intake
Evidence Level
Moderate
3 Human
5 Animal
2 In Vitro
Mechanism Leptin sensitization via amylin-mediated restoration of hypothalamic leptin responsiveness
Supported 4 direct studies
Benefit appears to overcome leptin resistance in obesity
Evidence Level
Moderate
1 Human
4 Animal
1 In Vitro
Mechanism Delayed gastric emptying via vagal efferent inhibition
Established 6 direct studies
Benefit shown to prolong satiety and reduce postprandial glucose spikes
Evidence Level
Moderate
2 Human
5 Animal
Mechanism Postprandial glucagon suppression via direct pancreatic alpha-cell effects
Supported 4 direct studies
Benefit appears to improve glycemic control in type 2 diabetes
Evidence Level
Moderate
2 Human
3 Animal
2 In Vitro
Mechanism Confidence
Established
Supported
Emerging
Evidence Level
High
Moderate
Low
Very Low
NCT ID Title Peptide Phase Status Completion
NCT03856047
Phase 2 Cagrilintide Monotherapy for Weight Management
Cagrilintide Phase 2 Completed Jan 2020
NCT04163354
Phase 1b Cagrilintide + Semaglutide Combination PK/PD
Cagrilintide Phase 1 Completed Jan 2020
NCT04940078
Phase 2 CagriSema in Type 2 Diabetes
Cagrilintide Phase 2 Completed Jan 2022
NCT05567796
REDEFINE 1: CagriSema vs Semaglutide in Obesity
Obesity
Cagrilintide Phase 3 Active Oct 2024
NCT05394519
REDEFINE 2: CagriSema in Obesity with T2D
Overweight, Obesity +1 more
Cagrilintide Phase 3 Completed Jan 2025
NCT06024720
REDEFINE 3: CagriSema vs Tirzepatide
Cagrilintide Phase 3 Active -
NCT05803421
REDEFINE CVOT: CagriSema Cardiovascular Outcomes
Cagrilintide Phase 3 Recruiting -
NCT07357740
A Research Study to Compare Two Different Versions of Injectable CagriSema in People With Type 2 Diabetes
Diabetes Mellitus, Type 2
Cagrilintide Phase 2 Not yet recruiting Aug 2027
NCT07282613
A Research Study to See How Much CagriSema Lowers Blood Sugar and Body Weight Compared to Placebo in Children and Adolescents With Type 2 Diabetes
Diabetes Mellitus, Type 2
Cagrilintide Phase 3 Not yet recruiting Sep 2029
NCT07589686
A Dose-Finding Study of Petrelintide With Enicepatide (RO7795068) in Adults With Obesity or Overweight
Obesity or Overweight
Cagrilintide Phase 2 Not yet recruiting Nov 2027
NCT07357766
A Research Study to Compare Different Versions of Injectable CagriSema and Placebo in People With Excess Body Weight
Overweight, Obesity
Cagrilintide Phase 3 Not yet recruiting Nov 2027
NCT07564414
A Research Study to Look at How Two Different Doses of CagriSema and One Dose of Semaglutide Help People Living With Obesity With or Without Type 2 Diabetes Lose Weight
Obesity, Type 2 Diabetes
Cagrilintide Phase 3 Recruiting Feb 2028
NCT07253285
A Research Study on How Well Cagrilintide and CagriSema Work in Children and Adolescents With Excess Body Weight
Overweight, Obesity
Cagrilintide Phase 3 Recruiting Mar 2030
NCT07220642
Weight Loss in People Living With Overweight or Obesity Following Treatment With Cagrilintide
Obesity, Overweight
Cagrilintide Phase 3 Active May 2027
NCT07220759
Weight Loss in People Living With Overweight or Obesity and Type 2 Diabetes Following Treatment With Cagrilintide
Overweight, Obesity +1 more
Cagrilintide Phase 3 Active May 2027
NCT07011667
A Research Study to Look at How Well CagriSema Helps People Living With Obesity Lose Weight and Maintain Weight Loss in the Long-term
Obesity
Cagrilintide Phase 3 Active Mar 2027
NCT06926842
Efficacy and Safety of Petrelintide in Participants With Overweight or Obesity and Type 2 Diabetes (ZUPREME 2)
Overweight, Type 2 Diabetes +1 more
Cagrilintide Phase 2 Active Aug 2026
NCT06951854
Phase II Clinical Trial to Evaluate the Efficacy and Safety of NV01-A02 in Children With Autism Spectrum Disorder
Autism Spectrum Disorder (ASD
Cagrilintide Phase 2 Recruiting Sep 2025
NCT06780449
A Research Study to Look Into the Long-term Effect on Weight Loss of CagriSema in People With Obesity
Obesity
Cagrilintide Phase 3 Active Aug 2028
NCT06797869
A Research Study to Investigate the Effects of CagriSema Compared to Placebo in People With Type 2 Diabetes and Painful Diabetic Peripheral Neuropathy
Diabetes Mellitus, Type 2, Diabetic Peripheral Neuropathy
Cagrilintide Phase 2 Active Aug 2026
NCT06534411
A Research Study to See How Much CagriSema Lowers Blood Sugar and Body Weight Compared to Tirzepatide in People With Type 2 Diabetes Treated With Metformin, SGLT2 Inhibitor or Both
Diabetes Mellitus, Type 2
Cagrilintide Phase 3 Active Jun 2026
NCT03856047 Completed

Phase 2 Cagrilintide Monotherapy for Weight Management

Cagrilintide Phase 2 Est. Jan 2020
NCT04163354 Completed

Phase 1b Cagrilintide + Semaglutide Combination PK/PD

Cagrilintide Phase 1 Est. Jan 2020
NCT04940078 Completed

Phase 2 CagriSema in Type 2 Diabetes

Cagrilintide Phase 2 Est. Jan 2022

REDEFINE 1: CagriSema vs Semaglutide in Obesity

Cagrilintide Phase 3 Est. Oct 2024
NCT05394519 Completed

REDEFINE 2: CagriSema in Obesity with T2D

Cagrilintide Phase 3 Est. Jan 2025

REDEFINE 3: CagriSema vs Tirzepatide

Cagrilintide Phase 3 Est. -
NCT05803421 Recruiting

REDEFINE CVOT: CagriSema Cardiovascular Outcomes

Cagrilintide Phase 3 Est. -
NCT07357740 Not yet recruiting

A Research Study to Compare Two Different Versions of Injectable CagriSema in People With Type 2 Diabetes

Cagrilintide Phase 2 Est. Aug 2027
NCT07282613 Not yet recruiting

A Research Study to See How Much CagriSema Lowers Blood Sugar and Body Weight Compared to Placebo in Children and Adolescents With Type 2 Diabetes

Cagrilintide Phase 3 Est. Sep 2029
NCT07589686 Not yet recruiting

A Dose-Finding Study of Petrelintide With Enicepatide (RO7795068) in Adults With Obesity or Overweight

Cagrilintide Phase 2 Est. Nov 2027
NCT07357766 Not yet recruiting

A Research Study to Compare Different Versions of Injectable CagriSema and Placebo in People With Excess Body Weight

Cagrilintide Phase 3 Est. Nov 2027
NCT07564414 Recruiting

A Research Study to Look at How Two Different Doses of CagriSema and One Dose of Semaglutide Help People Living With Obesity With or Without Type 2 Diabetes Lose Weight

Cagrilintide Phase 3 Est. Feb 2028
NCT07253285 Recruiting

A Research Study on How Well Cagrilintide and CagriSema Work in Children and Adolescents With Excess Body Weight

Cagrilintide Phase 3 Est. Mar 2030

Weight Loss in People Living With Overweight or Obesity Following Treatment With Cagrilintide

Cagrilintide Phase 3 Est. May 2027

Weight Loss in People Living With Overweight or Obesity and Type 2 Diabetes Following Treatment With Cagrilintide

Cagrilintide Phase 3 Est. May 2027

A Research Study to Look at How Well CagriSema Helps People Living With Obesity Lose Weight and Maintain Weight Loss in the Long-term

Cagrilintide Phase 3 Est. Mar 2027

Efficacy and Safety of Petrelintide in Participants With Overweight or Obesity and Type 2 Diabetes (ZUPREME 2)

Cagrilintide Phase 2 Est. Aug 2026
NCT06951854 Recruiting

Phase II Clinical Trial to Evaluate the Efficacy and Safety of NV01-A02 in Children With Autism Spectrum Disorder

Cagrilintide Phase 2 Est. Sep 2025

A Research Study to Look Into the Long-term Effect on Weight Loss of CagriSema in People With Obesity

Cagrilintide Phase 3 Est. Aug 2028

A Research Study to Investigate the Effects of CagriSema Compared to Placebo in People With Type 2 Diabetes and Painful Diabetic Peripheral Neuropathy

Cagrilintide Phase 2 Est. Aug 2026

A Research Study to See How Much CagriSema Lowers Blood Sugar and Body Weight Compared to Tirzepatide in People With Type 2 Diabetes Treated With Metformin, SGLT2 Inhibitor or Both

Cagrilintide Phase 3 Est. Jun 2026
Phase 01 1
Week 1-4

Initial titration period with dose escalation. Appetite suppression begins within days. GI side effects (nausea, vomiting) most common during this phase. Weight loss typically begins but is modest during titration.

PMID:34798060
Phase 02 2
Week 4-12

Continued weight loss as maintenance dose is reached. Mean weight loss of approximately 5-7% expected by week 12 based on Phase 2 trajectory. GI side effects typically improve after titration completion.

PMID:34798060
Phase 03 3
Week 12-26

Ongoing weight loss approaching plateau. Phase 2 monotherapy showed -10.8% at 26 weeks with cagrilintide 4.5 mg. Combination with semaglutide showed -17.1% at 20 weeks, projecting to greater efficacy with longer treatment.

PMID:33894838
Phase 04 4
Week 26+

Long-term maintenance phase. Phase 3 trials (REDEFINE) are 68 weeks duration. Weight loss plateau expected around week 40-68 based on GLP-1 agonist class data. Long-term efficacy and durability under investigation.

Research-based observations

This timeline reflects observations from published clinical and preclinical studies. Individual responses may vary significantly. This is not a guarantee of effects or a dosing schedule. Consult qualified healthcare providers for personalized guidance.

Good Signs (5 indicators)
Investigational compound - only available through clinical trials
Manufactured by Novo Nordisk under pharmaceutical-grade conditions
All published trial data from regulatory-grade clinical studies
Proper cold chain storage maintained
Clear documentation of trial enrollment
Warning Signs (4 indicators)
Any non-trial source claiming to sell cagrilintide
Products labeled as cagrilintide from research chemical suppliers
Claims of CagriSema availability outside clinical trials
Pricing significantly below pharmaceutical development costs
Bad Signs (5 indicators)
Cagrilintide sold online as research chemical (not legitimately available)
Any non-Novo Nordisk manufactured product
Claims of FDA approval (not yet approved as of January 2026)
Combination products from non-trial sources
Any product without proper pharmaceutical documentation
Positive quality indicator
Requires evaluation
Potential quality issue

For Research Evaluation Only

These quality indicators are general guidelines based on typical peptide characteristics. Professional laboratory testing (HPLC, mass spectrometry) provides definitive quality verification. This checklist is for initial visual evaluation only.

Synergistic
Compatible
Caution
Avoid

CagriSema is the combination product of cagrilintide + semaglutide. Phase 2 data shows -15.6% weight loss vs -5.1% for semaglutide alone. Complementary mechanisms via amylin and GLP-1 pathways.

Cagrilintide monotherapy showed comparable efficacy to liraglutide 3.0 mg in Phase 2. No specific interaction data but both can reduce appetite and slow gastric emptying.

Both are potent weight loss agents targeting distinct pathways. No combination studies exist. Concurrent use would have unknown safety profile and unclear benefit given overlapping GLP-1 receptor activity.

Research Note: Interaction data is based on published literature, mechanistic understanding, and theoretical considerations. Most peptide combinations lack direct clinical study. This information is for educational purposes only and does not constitute medical advice. Always consult qualified healthcare providers.

This dossier synthesizes available evidence from peer-reviewed literature, regulatory documents, and clinical trial registries. Evidence strength ratings follow a modified GRADE approach.

For complete methodology details, see our Methodology page.

Important Disclaimer

This dossier is for educational purposes only and does not constitute medical advice. Always consult a qualified healthcare provider before making health decisions.

Get Research Alerts

New dossiers and major study summaries delivered to your inbox. Evidence-graded, citation-backed research you can trust.

No spam. Unsubscribe anytime.

Compare Cagrilintide

Related Peptides

Metabolic

5-Amino-1MQ

5-Amino-1-Methylquinolinium · NNMT Inhibitor

A small molecule NNMT inhibitor studied for metabolic effects in animal models. No human clinical trials have been conducted. Increases NAD+ levels in adipose tissue in preclinical studies.

See dossier
Metabolic

Amycretin

NNC0487-0111 · Oral Amycretin · Subcutaneous Amycretin

A novel single-molecule dual GLP-1/amylin receptor agonist developed by Novo Nordisk. Unlike CagriSema (a fixed-dose combination), amycretin is a unified peptide that activates both pathways. Phase 1 trials showed superior weight loss signals versus semaglutide, with both oral and subcutaneous formulations in development.

See dossier
Metabolic

AOD-9604

Anti-Obesity Drug 9604 · Tyr-hGH Fragment 177-191 · hGH Fragment 176-191

A modified fragment of human growth hormone (amino acids 176-191 with N-terminal tyrosine) studied for fat loss. Clinical development discontinued after Phase 2b/3 trials failed to show efficacy in 536 subjects. Now prohibited by WADA and excluded from FDA compounding.

See dossier
Metabolic

CagriSema

Cagrilintide-Semaglutide · NNC0174-0833

A fixed-dose combination of cagrilintide (amylin analog) and semaglutide (GLP-1 agonist) for chronic weight management. Phase 3 REDEFINE trials demonstrate 20-23% weight loss at 68 weeks. NDA submitted to FDA December 2025. First GLP-1/amylin combination therapy.

See dossier
Metabolic

CT-388

RG-6912

A dual GLP-1/GIP receptor agonist (INN enicepatide; also RO7795068) acquired by Roche through the $2.7 billion Carmot Therapeutics acquisition in 2024. The published Phase 1 trial (NCT04838405) showed 4.7-8.0% mean weight loss vs 0.5% placebo over 4 weeks; a more widely reported ~18.8% placebo-adjusted figure at 24 weeks comes from an unpublished Phase 1 extension reported via press release. Phase 2 obesity and T2D trials are completed or ongoing and Phase 3 began in 2026, positioning it as a competitive obesity therapeutic with a mechanism similar to tirzepatide.

See dossier
Metabolic

Ecnoglutide

XW003 · Sciwind GLP-1

A long-acting GLP-1 receptor agonist developed by Sciwind Biosciences. A Phase 3 obesity trial showed 13.2% weight loss at 40 weeks with once-weekly dosing. Primarily targeting China and Asian markets with potential for global expansion.

See dossier

Related Content